SCHEMBL15313754

SCHEMBL15313754

NS(=O)(=O)c1ccc(CCNS(=O)(=O)c2ccc3c(c2)CN(C(=O)c2cc(S(=O)(=O)N4CCc5ccccc5C4)c(O)c(O)c2O)CC3)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 3/20 0.65
MCL1 Q07820 1/20 0.63
BAD Q92934 1/20 0.63
CA1 P00915 4/20 0.45
CA2 P00918 4/20 0.45
CA7 P43166 3/20 0.45
CA9 Q16790 3/20 0.45
CA14 Q9ULX7 3/20 0.45
LMNA P02545 4/20 0.42
ALDH1A1 P00352 4/20 0.42
HTT P42858 3/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
BACE1 P56817 1/20 0.42
MAPK1 P28482 3/20 0.41
AKR1C3 P42330 1/20 0.41
KMT2A Q03164 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15313742 0.94 BCL2 (0.73) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313753 0.93 BCL2 (0.65) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313763 0.93 BCL2 (0.67) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313961 0.91 BCL2 (0.65) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313756 0.91 BCL2 (0.65) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313757 0.89 BCL2 (0.69) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313751 0.88 BCL2 (0.63) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313762 0.88 BCL2 (0.59) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313755 0.87 BCL2 (0.64) BCL2MCL1BADLMNAALDH1A1
SCHEMBL15313741 0.86 BCL2 (0.61) BCL2MCL1BADLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed