SCHEMBL15327367

SCHEMBL15327367

CC1(C(=O)N2C[C@H](S(=O)(=O)c3ccc(OCC(F)(F)F)cc3Cl)C[C@@H]2OC(=O)NC2(C#N)CC2)COC1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSS P25774 20/20 0.59
CTSL P07711 18/20 0.59
CTSK P43235 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15327277 0.94 CTSS (0.62) CTSSCTSLCTSK
SCHEMBL15327313 0.90 CTSS (0.63) CTSSCTSLCTSK
SCHEMBL694472 0.90 CTSS (0.73) CTSSCTSLCTSK
SCHEMBL15327407 0.89 CTSS (0.62) CTSSCTSL
SCHEMBL15327523 0.89 CTSS (0.62) CTSSCTSL
SCHEMBL15327372 0.89 CTSS (0.61) CTSSCTSLCTSK
SCHEMBL15327395 0.88 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL15327567 0.87 CTSL (0.60) CTSSCTSLCTSK
SCHEMBL15327413 0.87 CTSS (0.52) CTSSCTSL
SCHEMBL15327549 0.87 CTSL (0.63) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-B1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS HOFFMANN LA ROCHE (CH) 2013-10-23 EP claimed