SCHEMBL15330666

SCHEMBL15330666

O=Cc1ccc(N2CCNC(=O)CC2)c(F)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.62
SMN1; SMN2 Q16637 3/20 0.62
ALDH1A3 P47895 6/20 0.42
MAPT P10636 5/20 0.41
MITF O75030 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 3/20 0.40
ALDH3A1 P30838 1/20 0.40
MEN1 O00255 2/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM1A O60341 1/20 0.34
PIK3CA P42336 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2560082 0.88 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2ALDH1A3MAPTMITF
SCHEMBL15330735 0.85 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2MAPTPIK3CAPARP1
SCHEMBL15332950 0.84 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2ALDH1A3MAPTHTT
SCHEMBL4934676 0.83 ALDH1A1 (0.73) ALDH1A1SMN1; SMN2ALDH1A3MAPTMITF
SCHEMBL31494990 0.83 ALDH1A1 (0.73) ALDH1A1SMN1; SMN2ALDH1A3MAPTMITF
Hydrochloric Acid SCHEMBL29952847 0.81 ALDH1A1 (0.71) ALDH1A1SMN1; SMN2ALDH1A3MAPTMITF
SCHEMBL22542024 0.81 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2MAPTHTTKMT2A
SCHEMBL5246344 0.81 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2MAPTHTTKMT2A
SCHEMBL15329506 0.80 ALDH1A1 (0.66) ALDH1A1SMN1; SMN2ALDH1A3MAPTHTT
SCHEMBL20883567 0.78 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed