SCHEMBL1534443

SCHEMBL1534443

O=c1c(I)c(-c2ccccc2)oc2c(=O)n(CCO)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.37
KDM4E B2RXH2 4/20 0.35
CYP3A4 P08684 3/20 0.35
LMNA P02545 2/20 0.35
ACHE P22303 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
CHRM2 P08172 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CHRM1 P11229 1/20 0.35
SLC6A2 P23975 1/20 0.35
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1534503 0.86 ALDH1A1 (0.39) ABCG2KDM4ECYP3A4LMNAACHE
SCHEMBL1534597 0.81 ABCG2 (0.39) ABCG2KDM4ECYP3A4LMNAACHE
SCHEMBL1534935 0.75 AKT1 (0.41)
Hydrochloric Acid SCHEMBL1534506 0.74 AKT1 (0.40)
SCHEMBL1534620 0.73 ABCG2 (0.40) ABCG2KDM4ECYP3A4LMNAACHE
SCHEMBL1534696 0.73 ABCG2 (0.40) ABCG2KDM4ECYP3A4LMNAACHE
SCHEMBL1534677 0.71 ABCG2 (0.35) ABCG2KDM4ECYP3A4LMNAACHE
SCHEMBL1534801 0.69 ABCG2 (0.51) ABCG2KDM4ECYP3A4LMNAACHE
SCHEMBL1534426 0.68 ABCG2 (0.43) ABCG2KDM4ECYP3A4LMNACYP1A2
SCHEMBL1534523 0.68 ABCG2 (0.43) ABCG2KDM4ECYP3A4LMNAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8546376-B2 Pharmaceutical compounds ALMAC DISCOVERY LIMITED (GB) 2013-10-01 US disclosed
US-20120238541-A1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2012-09-20 US disclosed
EP-2473495-A1 PHARMACEUTICAL COMPOUNDS Almac Discovery Limited (GB) 2012-07-11 EP disclosed
WO-2011033265-A1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2011-03-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120238541-A1 PHARMACEUTICAL COMPOUNDS PIK3CA, PLK1, MTOR ABCG2 507/4885KDM4E 1952/4885CYP3A4 2648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.