SCHEMBL1534518

SCHEMBL1534518

O=C(O)NC1(c2ccc(-c3c(-c4ccccc4)oc4ccc(F)cc4c3=O)cc2)CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
CYP2C8 P10632 3/20 0.46
MAPK14 Q16539 6/20 0.43
PLA2G2A P14555 1/20 0.43
PLA2G4A P47712 1/20 0.43
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SCN9A Q15858 1/20 0.41
PIK3CD O00329 1/20 0.40
PIK3R2 O00459 1/20 0.40
PIK3CG P48736 1/20 0.40
TNKS O95271 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1534320 0.88 CYP3A4 (0.42) CYP3A4CYP2C8MAPK14PLA2G2APLA2G4A
SCHEMBL1534546 0.83 PLA2G2A (0.42) CYP3A4CYP2C8MAPK14PLA2G2APLA2G4A
SCHEMBL14118764 0.83 TACR3 (0.42) CYP3A4CYP2C8MAPK14PLA2G2APLA2G4A
SCHEMBL1534389 0.82 MAPK14 (0.47) MAPK14PLA2G2APLA2G4ATNKS
SCHEMBL1534850 0.81 AKT1 (0.42) CYP3A4CYP2C8MAPK14PLA2G2APLA2G4A
SCHEMBL1900240 0.80 VNN1 (0.41) CYP3A4CYP2C8PLA2G2APLA2G4AKDM4E
SCHEMBL14119098 0.80 IP6K1 (0.43) CYP3A4CYP2C8PLA2G2APLA2G4AKDM4E
SCHEMBL1534621 0.79 AKT1 (0.42) CYP3A4CYP2C8MAPK14PLA2G2APLA2G4A
SCHEMBL1534823 0.78 TACR3 (0.37) CYP3A4MAPK14PLA2G2APLA2G4AKDM4E
SCHEMBL1534471 0.78 AKT1 (0.45) CYP3A4CYP2C8PLA2G2APLA2G4AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473495-A1 PHARMACEUTICAL COMPOUNDS Almac Discovery Limited (GB) 2012-07-11 EP disclosed
WO-2011033265-A1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2011-03-24 WO disclosed