SCHEMBL15375665

SCHEMBL15375665

CCOC(C)c1ccc(C#Cc2ccc(C(=O)N[C@H](C(=O)OC)[C@@H](C)NC(=O)OCC3c4ccccc4-c4ccccc43)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.38
CASP3 P42574 3/20 0.37
TLR2 O60603 4/20 0.37
PIN1 Q13526 1/20 0.36
ACACB O00763 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3012552 0.90 CASP3 (0.43) KMT2ACASP3PIN1
SCHEMBL3018948 0.87 KMT2A (0.43) KMT2ACASP3PIN1
SCHEMBL3808020 0.87 KMT2A (0.43) KMT2ACASP3PIN1
SCHEMBL3018189 0.87 ACACB (0.40) KMT2ACASP3TLR2PIN1ACACB
SCHEMBL3018006 0.86 KMT2A (0.40) KMT2ACASP3PIN1ACACB
SCHEMBL3008053 0.85 CASP3 (0.41) KMT2ACASP3PIN1
SCHEMBL3015812 0.85 KMT2A (0.44) KMT2ACASP3TLR2PIN1ACACB
SCHEMBL13984775 0.85 CASP3 (0.41) KMT2ACASP3PIN1
SCHEMBL3802721 0.85 KMT2A (0.44) KMT2ACASP3TLR2PIN1ACACB
SCHEMBL15375666 0.85 ACACB (0.39) KMT2ACASP3TLR2PIN1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2662353-A2 Antibacterial agents Achaogen, Inc. (US) 2013-11-13 EP disclosed