SCHEMBL15404591

SCHEMBL15404591

CN(C)C(=O)[C@H]1C[C@H](NC(=O)O)C1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MME P08473 2/20 0.35
DPP4 P27487 1/20 0.34
FASN P49327 3/20 0.32
ATM Q13315 1/20 0.31
PDE7A Q13946 2/20 0.31
PPM1B O75688 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15404590 1.00 MME (0.35) MMEDPP4FASNATMPDE7A
SCHEMBL22042454 0.91 MME (0.32) MMEDPP4
SCHEMBL22042599 0.91 MME (0.32) MMEDPP4
SCHEMBL22042408 0.89 MME (0.31) MME
SCHEMBL14658519 0.83 MME (0.46) MMEFASNPDE7A
SCHEMBL3715481 0.83 MME (0.46) MMEFASNPDE7A
SCHEMBL7447161 0.83 MME (0.50) MMEDPP4FASNPDE7ATSHR
SCHEMBL22042484 0.81 MMP2 (0.33)
SCHEMBL23826739 0.80 CHRNB2 (0.32)
SCHEMBL16240628 0.80 CHRNB2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684880-B1 DISPIROPYRROLIDINE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2018-02-28 EP disclosed
US-20140121196-A1 DISPIROPYRROLIDINE DERIVATIVES DAIICHI SANKYO COMPANY, LIMITED (JP) 2014-05-01 US disclosed
EP-2684880-A1 DISPIROPYRROLIDINE DERIVATIVE DAIICHI SANKYO COMPANY, LIMITED (JP) 2014-01-15 EP disclosed
US-8629133-B2 Dispiropyrrolidine derivatives DAIICHI SANKYO COMPANY, LIMITED (JP) 2014-01-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140121196-A1 DISPIROPYRROLIDINE DERIVATIVES MDM2, TP53, TPD52L2 MME 4106/4885DPP4 2001/4885FASN 4688/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.