Formic Acid

Formic Acid

SCHEMBL15411803

Cc1c(-c2ccnn2-c2ccc(C#N)cc2)cn2nc(NC(=O)NCCC[N+](C)(C)C)nc2c1-c1cccc(C(F)(F)F)c1.O=C[O-]

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ELANE P08246 7/20 0.41
EPHX2 P34913 7/20 0.37
PTGS2 P35354 7/20 0.37
AKR1C3 P42330 1/20 0.33
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
MALT1 Q9UDY8 1/20 0.32
ADORA2A P29274 1/20 0.32
SLC5A1 P13866 2/20 0.32
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL15411805 0.98 ELANE (0.42) ELANEEPHX2PTGS2AKR1C3ITGB2
SCHEMBL15425453 0.97 ELANE (0.43) ELANEEPHX2PTGS2AKR1C3ITGB2
Formic Acid SCHEMBL15411865 0.94 ELANE (0.39) ELANEEPHX2PTGS2AKR1C3ITGB2
Formic Acid SCHEMBL15411868 0.91 ELANE (0.40) ELANEEPHX2PTGS2AKR1C3ITGB2
SCHEMBL15425553 0.91 ELANE (0.41) ELANEEPHX2PTGS2AKR1C3ITGB2
SCHEMBL15411853 0.90 ELANE (0.44) ELANEEPHX2PTGS2ITGB2ICAM1
SCHEMBL15410928 0.90 ELANE (0.45) ELANEEPHX2PTGS2AKR1C3ITGB2
Formic Acid SCHEMBL15411730 0.90 ELANE (0.41) ELANEMALT1ADORA2ASLC5A1MAPT
Formic Acid SCHEMBL15412289 0.90 ELANE (0.41) ELANE
SCHEMBL15411653 0.89 ELANE (0.43) ELANEEPHX2PTGS2ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2872509-B1 INHIBITION OF ENZYMES CHIESI FARMA SPA (IT) 2016-09-14 EP claimed
US-9199984-B2 Inhibition of enzymes CHIESI FARMACEUTICI S.P.A. (IT) 2015-12-01 US claimed
EP-2872509-A1 INHIBITION OF ENZYMES Chiesi Farmaceutici S.p.A. (IT) 2015-05-20 EP claimed
WO-2014009425-A1 INHIBITION OF ENZYMES CHIESI FARMACEUTICI S.P.A. (IT) 2014-01-16 WO claimed
US-20140018345-A1 INHIBITION OF ENZYMES CHIESI FARMACEUTICI S.P.A (IT) 2014-01-16 US claimed
EP-2872509-B1 INHIBITION OF ENZYMES CHIESI FARMA SPA (IT) 2016-09-14 EP disclosed
US-9199984-B2 Inhibition of enzymes CHIESI FARMACEUTICI S.P.A. (IT) 2015-12-01 US disclosed
EP-2872509-A1 INHIBITION OF ENZYMES Chiesi Farmaceutici S.p.A. (IT) 2015-05-20 EP disclosed
WO-2014009425-A1 INHIBITION OF ENZYMES CHIESI FARMACEUTICI S.P.A. (IT) 2014-01-16 WO disclosed
US-20140018345-A1 INHIBITION OF ENZYMES CHIESI FARMACEUTICI S.P.A (IT) 2014-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140018345-A1 INHIBITION OF ENZYMES SERPINB1, ELANE, MPO ELANE 2/4885EPHX2 473/4885PTGS2 684/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.