Acridan

Acridan

SCHEMBL15412652

N.c1ccc2c(c1)Cc1ccccc1N2

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.62
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
NPC1 O15118 2/20 0.62
KDM4E B2RXH2 2/20 0.62
AHR P35869 1/20 0.62
PDK2 Q15119 1/20 0.62
HSP90AA1 P07900 1/20 0.62
THRB P10828 1/20 0.62
HK1 P19367 1/20 0.62
MAPK1 P28482 1/20 0.62
RECQL P46063 1/20 0.62
RAB9A P51151 1/20 0.62
GALK1 P51570 1/20 0.62
BLM P54132 1/20 0.62
HKDC1 Q2TB90 1/20 0.62
ALOX15 P16050 2/20 0.56
HSD17B10 Q99714 1/20 0.56
BRD4 O60885 2/20 0.48
CREBBP Q92793 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridan SCHEMBL29446489 0.97 MAPT (0.65) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL20594012 0.97 MAPT (0.65) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL183367 0.97 MAPT (0.65) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL29405807 0.97 MAPT (0.65) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL28832553 0.94 MAPT (0.62) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL29006126 0.94 MAPT (0.62) MAPTMEN1KMT2ANPC1KDM4E
SCHEMBL4571016 0.94 MAPT (0.62) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL29020974 0.94 MAPT (0.62) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL10813635 0.94 MAPT (0.62) MAPTMEN1KMT2ANPC1KDM4E
Acridan SCHEMBL28268824 0.94 MAPT (0.62) MAPTMEN1KMT2ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104411688-B Synthesis of acridinium compounds from N-alkylation of 9,10-dihydroacridine 西门子医疗保健诊断公司 2019-01-08 CN disclosed
EP-2872489-B1 SYNTHESIS OF ACRIDINIUM COMPOUNDS BY N-ALKYLATION OF ACRIDANS SIEMENS HEALTHCARE DIAGNOSTICS INC (US) 2016-12-21 EP disclosed
US-9512080-B2 Synthesis of acridinium compounds by N-alkylation of acridans SIEMENS HEALTHCARE DIAGNOSTICS INC. (US) 2016-12-06 US disclosed
US-20150197491-A1 SYNTHESIS OF ACRIDINIUM COMPOUNDS BY N-ALKYLATION OF ACRIDANS SIEMENS HEALTHCARE DIAGNOSTICS INC. (US) 2015-07-16 US disclosed
EP-2872489-A1 SYNTHESIS OF ACRIDINIUM COMPOUNDS BY N-ALKYLATION OF ACRIDANS Siemens Healthcare Diagnostics Inc. (US) 2015-05-20 EP disclosed
WO-2014011762-A1 SYNTHESIS OF ACRIDINIUM COMPOUNDS BY N-ALKYLATION OF ACRIDANS SIEMENS HEAL THCARE DIAGNOSTICS INC. (US) 2014-01-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150197491-A1 SYNTHESIS OF ACRIDINIUM COMPOUNDS BY N-ALKYLATION OF ACRIDANS ACR, MCL1, MGMT MAPT 4190/4885MEN1 983/4885KMT2A 1929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.