SCHEMBL15418951

SCHEMBL15418951

Cn1c(=O)c(C(=O)NC(C(=O)O)C(C)(C)C)c(O)c2ccc(Br)cc21

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.64
L3MBTL1 Q9Y468 1/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
GAA P10253 1/20 0.48
GSK3B P49841 2/20 0.45
HIF1A Q16665 11/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2382306 0.86 EGLN1 (0.67) EGLN1L3MBTL1MEN1KMT2AGAA
SCHEMBL2382301 0.86 EGLN1 (0.67) EGLN1L3MBTL1MEN1KMT2AGAA
SCHEMBL12254437 0.82 EGLN1 (0.64) EGLN1L3MBTL1MEN1KMT2AGAA
SCHEMBL15419072 0.81 L3MBTL1 (0.44) EGLN1L3MBTL1MEN1KMT2AHIF1A
SCHEMBL15419045 0.81 EGLN1 (0.68) EGLN1L3MBTL1MEN1KMT2AGAA
SCHEMBL15419070 0.81 L3MBTL1 (0.45) EGLN1L3MBTL1MEN1KMT2AHIF1A
SCHEMBL2385032 0.80 EGLN1 (0.61) EGLN1L3MBTL1MEN1KMT2AGAA
SCHEMBL2385033 0.80 EGLN1 (0.61) EGLN1L3MBTL1MEN1KMT2AGAA
SCHEMBL2384498 0.78 EGLN1 (1.00) EGLN1HIF1A
SCHEMBL15419151 0.77 GSK3B (0.56) EGLN1L3MBTL1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960363-B1 QUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS AND USES THEREOF AMGEN INC (US) 2014-01-22 EP claimed