SCHEMBL15424419

SCHEMBL15424419

[N-]=[N+]=N[C@H]1CO[C@@H]2COC(c3ccccc3)CC[C@H]2C1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15424384 0.75 TSHR (0.47) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL13453023 0.74 ALDH1A1 (0.38) TSHR
SCHEMBL24311520 0.74 ALDH1A1 (0.38) TSHR
SCHEMBL13771105 0.74 ALDH1A1 (0.38) TSHR
SCHEMBL17029485 0.74 TSHR (0.40) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL13934947 0.70 MEN1 (0.44) TSHR
SCHEMBL5072064 0.64 TSHR (0.55) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL25947955 0.63 TSHR (0.50) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL14336754 0.63 SLC18A3 (0.44) TSHR
SCHEMBL21026 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684880-A1 DISPIROPYRROLIDINE DERIVATIVE DAIICHI SANKYO COMPANY, LIMITED (JP) 2014-01-15 EP disclosed