SCHEMBL15426465

SCHEMBL15426465

Cc1cnc2c(c1)nc(-c1ccccc1F)n2C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.41
PDE10A Q9Y233 6/20 0.40
PDE2A O00408 3/20 0.40
AKT1 P31749 2/20 0.40
AKT2 P31751 2/20 0.40
BRD4 O60885 1/20 0.40
MBNL1 Q9NR56 1/20 0.39
CYP1A2 P05177 1/20 0.39
NPC1 O15118 2/20 0.39
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.38
GRM2 Q14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15426501 0.89 HSD11B1 (0.42) HSD11B1PDE10APDE2AAKT1AKT2
SCHEMBL15426510 0.84 BRD4 (0.40) PDE10ABRD4CYP1A2
SCHEMBL15426491 0.84 AKT1 (0.38) PDE10APDE2AAKT1AKT2BRD4
SCHEMBL9953426 0.84 PDE2A (0.49) HSD11B1PDE10APDE2AMBNL1
SCHEMBL15426503 0.83 GRIN2B (0.43) PDE10AAKT1AKT2BRD4CYP1A2
SCHEMBL10248903 0.83 POLB (0.38) PDE10AAKT1AKT2CYP11B2CYP11B1
SCHEMBL15426254 0.82 KDM4E (0.39) PDE10APDE2AAKT1AKT2BRD4
SCHEMBL15868287 0.81 AKT1 (0.41) PDE10AAKT1AKT2BRD4NPC1
SCHEMBL15426486 0.80 HSD11B1 (0.47) HSD11B1PDE10APDE2ACYP1A2CYP11B2
SCHEMBL15426495 0.80 ALDH1A1 (0.40) PDE10AAKT1AKT2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9278983-B2 Fused heterocyclic compound and use thereof for pest control SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2016-03-08 US disclosed
US-20140364444-A1 FUSED HETEROCYCLIC COMPOUND AND USE THEREOF FOR PEST CONTROL SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2014-12-11 US disclosed
US-8853238-B2 Fused heterocyclic compound and use thereof for pest control SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2014-10-07 US disclosed
US-20140018373-A1 FUSED HETEROCYCLIC COMPOUND AND USE FOR PEST CONTROL THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2014-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140018373-A1 FUSED HETEROCYCLIC COMPOUND AND USE FOR PEST CONTROL THEREOF NR4A1, NR2C2, NR0B1 HSD11B1 1704/4885PDE10A 3812/4885PDE2A 3467/4885
US-20140364444-A1 FUSED HETEROCYCLIC COMPOUND AND USE THEREOF FOR PEST CONTROL NR4A1, NR2C2, NR0B1 HSD11B1 1639/4885PDE10A 3725/4885PDE2A 3420/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.