SCHEMBL15428850

SCHEMBL15428850

O=C(O)c1ccc(-c2ccc(-c3ccc4cc[nH]c4c3)cn2)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ENPP2 Q13822 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM4C Q9H3R0 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
CHRNA7 P36544 2/20 0.38
KCNH2 Q12809 2/20 0.38
PIM1 P11309 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
MCL1 Q07820 1/20 0.37
ABL1 P00519 1/20 0.37
PTPN1 P18031 1/20 0.37
PIK3CD O00329 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15428851 0.91 NPC1 (0.43) ALDH1A1HPGDENPP2CCNCCDK8
SCHEMBL3377274 0.84 ALDH1A1 (0.51) ALDH1A1HPGDKDM4EENPP2HSD17B10
SCHEMBL1299857 0.83 ALDH1A1 (0.41) ALDH1A1HPGDKDM4EENPP2HSD17B10
SCHEMBL1316087 0.79 MMP13 (0.47)
SCHEMBL3413733 0.77 ALDH1A1 (0.66) ALDH1A1HPGDKDM4ENR4A1NR4A2
SCHEMBL1317504 0.76 NR4A1 (0.68) ALDH1A1HPGDNR4A1NR4A2NR4A3
SCHEMBL1317581 0.75 NR4A1 (0.56) ALDH1A1HPGDKDM4ENR4A1NR4A2
SCHEMBL1317461 0.75 NR4A1 (0.51) ALDH1A1HPGDKDM4ENR4A1NR4A2
SCHEMBL1317391 0.75 ALDH1A1 (0.46) ALDH1A1HPGDKDM4ENR4A1NR4A2
SCHEMBL1319813 0.75 ALDH1A1 (0.50) ALDH1A1HPGDKDM4ENR4A1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637550-B2 Heteroaryl diamide compounds useful as MMP-13 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-28 US disclosed