SCHEMBL1542886

SCHEMBL1542886

O=C(O)/C=C/C(=O)Oc1c(-c2ccc(OC3CN4CCC3CC4)cc2)[nH]c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
LSS P48449 1/20 0.42
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3192106 0.96 CHRNA7 (0.45) CHRNA7HTR3EHTR3BCHRNB2CHRNA4
Fumaric Acid SCHEMBL3192099 0.78 LSS (0.44) LSS
Fumaric Acid SCHEMBL1542888 0.78 LSS (0.44) LSS
Fumaric Acid SCHEMBL5420562 0.76 CHRNA7 (0.50) CHRNA7LSSBCHEACHECHRM2
Fumaric Acid SCHEMBL5420571 0.76 CHRNA7 (0.50) CHRNA7LSSBCHEACHECHRM2
Fumaric Acid SCHEMBL1542469 0.76 GYS1 (0.46) CHRNA7HTR3EHTR3BCHRNB2CHRNA4
Fumaric Acid SCHEMBL1542464 0.76 GYS1 (0.46) CHRNA7HTR3EHTR3BCHRNB2CHRNA4
Fumaric Acid SCHEMBL1020193 0.74 LSS (0.53) CHRNA7LSSBCHEACHEMEN1
SCHEMBL5650254 0.74 LSS (0.57) CHRNA7LSSBCHEACHEMEN1
SCHEMBL5420568 0.72 CHRM2 (0.50) CHRNA7LSSBCHEACHECHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2308875-A1 Fused bicycloheterocycle substituted quinuclidine derivatives as .alpha.7 nAChR modulators Abbott Laboratories (US) 2011-04-13 EP disclosed