SCHEMBL15428862

SCHEMBL15428862

N#Cc1ccc(C(=O)NCc2cccc(-c3ccc(C(=O)O)o3)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.57
EPHX2 P34913 3/20 0.50
MAOA P21397 2/20 0.48
IDO1 P14902 1/20 0.48
KDM1A O60341 1/20 0.47
HDAC1 Q13547 1/20 0.47
PPARA Q07869 1/20 0.47
RAB9A P51151 1/20 0.47
NR1H4 Q96RI1 2/20 0.46
NR4A1 P22736 1/20 0.46
NR4A2 P43354 1/20 0.46
NR4A3 Q92570 1/20 0.46
KCNH2 Q12809 1/20 0.46
SCN10A Q9Y5Y9 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK2 O75116 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15428855 0.90 CHRM3 (0.57) CHRM3EPHX2MAOANR1H4NR4A1
SCHEMBL1318756 0.87 NR1H4 (0.55) EPHX2NR1H4NR4A1NR4A2NR4A3
SCHEMBL15428849 0.85 MMP13 (0.54) EPHX2RAB9ANR1H4NR4A1NR4A2
SCHEMBL15428870 0.83 KMT2A (0.67) CHRM3EPHX2RAB9ANR1H4KMT2A
SCHEMBL15428868 0.83 SMN1; SMN2 (0.53) EPHX2RAB9ANR1H4NR4A1NR4A2
SCHEMBL15428860 0.83 KDM4E (0.53) CHRM3EPHX2HDAC1NR1H4NR4A1
SCHEMBL1317297 0.82 CHRM3 (0.59) CHRM3EPHX2MAOAIDO1KDM1A
SCHEMBL15428856 0.81 NR1H4 (0.60) EPHX2RAB9ANR1H4NR4A1NR4A2
SCHEMBL1318959 0.81 MMP13 (0.63) CHRM3
SCHEMBL15428864 0.80 MMP13 (0.65) CHRM3KMT2AROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637550-B2 Heteroaryl diamide compounds useful as MMP-13 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-28 US disclosed