SCHEMBL15428875

SCHEMBL15428875

CNC(=O)[CH][C@@H](C)CC(N)=O

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
ECE1 P42892 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15428858 1.00 CHRNB2 (0.35) CHRNB2CHRNB4CHRNA3CHRNA4ECE1
SCHEMBL3661088 0.83 ECE1 (0.33) ECE1
SCHEMBL3695948 0.82 ECE1 (0.32) ECE1
SCHEMBL3667412 0.80 ECE1 (0.34) ECE1
SCHEMBL3661960 0.80 ECE1 (0.31) ECE1
SCHEMBL3665726 0.79 ECE1 (0.30) ECE1
SCHEMBL2142444 0.78 ECE1 (0.32) ECE1
SCHEMBL5049589 0.78 ECE1 (0.32) ECE1
SCHEMBL3666706 0.77 ECE1 (0.36) CHRNB2CHRNB4CHRNA3CHRNA4ECE1
SCHEMBL3663065 0.77 ALOX15 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346831-B1 HETEROARYL DIAMIDE COMPOUNDS USEFUL AS MMP-13 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2015-01-07 EP disclosed
US-8637550-B2 Heteroaryl diamide compounds useful as MMP-13 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-28 US disclosed