SCHEMBL15428879

SCHEMBL15428879

CN(C)c1cccc(C(=O)NCc2cccc(-c3ccc(C(=O)O)o3)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.58
CHRM3 P20309 1/20 0.56
KDM4E B2RXH2 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 2/20 0.48
TMEM97 Q5BJF2 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
MMP13 P45452 3/20 0.47
EPHX2 P34913 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
ROCK2 O75116 2/20 0.47
ROCK1 Q13464 2/20 0.47
CFD P00746 1/20 0.46
RPA1 P27694 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NR4A1 P22736 1/20 0.45
NR4A2 P43354 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15428860 0.90 KDM4E (0.53) POLBCHRM3KDM4ESMN1; SMN2MMP13
SCHEMBL1318756 0.86 NR1H4 (0.55) KDM4ESMN1; SMN2LMNAMMP13EPHX2
SCHEMBL15428857 0.86 CHRM3 (0.54) POLBCHRM3LMNAMMP13EPHX2
SCHEMBL15428864 0.84 MMP13 (0.65) CHRM3LMNAMMP13ROCK2ROCK1
SCHEMBL15428881 0.83 PPARG (0.49) LMNAMMP13EPHX2NR1H4CFD
SCHEMBL1317689 0.83 CHRM3 (0.58) POLBCHRM3KDM4ESMN1; SMN2LMNA
SCHEMBL15428856 0.83 NR1H4 (0.60) KDM4ESMN1; SMN2MMP13EPHX2NR1H4
SCHEMBL7918709 0.82 MMP13 (0.63) POLBCHRM3MMP13
SCHEMBL1316491 0.82 MMP13 (0.63) POLBCHRM3MMP13
SCHEMBL15428849 0.82 MMP13 (0.54) POLBSMN1; SMN2LMNATP53MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637550-B2 Heteroaryl diamide compounds useful as MMP-13 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-28 US disclosed