SCHEMBL15434244

SCHEMBL15434244

CN/C=C/C(=O)c1cn2nc(NC(C)=O)nc2c(-c2cccc(C(F)(F)F)c2)c1C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.40
ALDH1A1 P00352 2/20 0.38
PIK3CG P48736 6/20 0.37
PIK3CD O00329 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MC4R P32245 1/20 0.37
TOP2A P11388 1/20 0.36
FYN P06241 1/20 0.36
PIK3CB P42338 2/20 0.36
JAK2 O60674 1/20 0.36
NPY5R Q15761 3/20 0.35
TLR7 Q9NYK1 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
MAT2A P31153 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15411539 0.89 ALDH1A1 (0.43) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15411537 0.89 ALDH1A1 (0.43) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15411158 0.88 ADORA2A (0.45) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15411630 0.86 ADORA2A (0.44) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15411350 0.84 ADORA2A (0.42) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15410377 0.82 ADORA2A (0.45) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15411621 0.82 ADORA2A (0.39) ADORA2AALDH1A1PIK3CGPIK3CDSMN1; SMN2
SCHEMBL15411069 0.74 EGLN2 (0.42) ADORA2APIK3CGPIK3CDMC4RTOP2A
SCHEMBL18076251 0.73 MALT1 (0.40) ADORA2AALDH1A1PIK3CGPIK3CDTOP2A
SCHEMBL15410874 0.73 EGLN2 (0.40) ADORA2AALDH1A1MC4RTOP2AFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014009425-A1 INHIBITION OF ENZYMES CHIESI FARMACEUTICI S.P.A. (IT) 2014-01-16 WO disclosed