SCHEMBL15435532

SCHEMBL15435532

CCOC(=O)c1c(Br)c(C#N)n(COCC[SiH2]C)c1Br

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.34
ALDH1A1 P00352 7/20 0.33
KDM4E B2RXH2 3/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 1/20 0.32
HTT P42858 2/20 0.30
USP2 O75604 1/20 0.30
LMNA P02545 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
RAD52 P43351 1/20 0.30
PKM P14618 1/20 0.30
CCR6 P51684 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL275025 0.84 ALDH1A1 (0.34) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL14493863 0.82 ALDH1A1 (0.33) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10225364 0.68 NPC1 (0.31)
SCHEMBL24553235 0.62 KDM4E (0.47) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL275429 0.61 DGAT1 (0.38) MAPTALDH1A1KDM4EHSD17B10HTT
SCHEMBL11563077 0.59 MAPT (0.52) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL13217488 0.59 KDM4E (0.43) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL28999329 0.57 HPGD (0.41) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL17165495 0.57 SMN1; SMN2 (0.48) MAPTALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11008658 0.56 ALDH1A1 (0.62) MAPTALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957077-B1 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC (US) 2014-01-22 EP disclosed