Xylazine

Xylazine

SCHEMBL15487

Cc1cccc(C)c1NC1=NCCCS1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 1.00
CYP3A4 P08684 1/20 1.00
CYP2D6 P10635 1/20 1.00
TSHR P16473 1/20 1.00
RAB9A P51151 1/20 1.00
MAPT P10636 1/20 0.97
BLM P54132 1/20 0.97
PMP22 Q01453 1/20 0.97
SMN1; SMN2 Q16637 2/20 0.69
GAA P10253 2/20 0.57
ALDH1A1 P00352 2/20 0.57
POLB P06746 2/20 0.51
KMT2A Q03164 3/20 0.49
HTR1D P28221 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xylazine SCHEMBL38986 0.98 LMNA (1.00) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL1119093 0.98 LMNA (1.00) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL22616146 0.98 LMNA (0.97) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL18988891 0.98 LMNA (0.97) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL1228390 0.98 LMNA (1.00) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL3339638 0.97 LMNA (0.94) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL9808825 0.91 LMNA (0.83) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL22616203 0.91 RAB9A (0.83) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL22616197 0.91 LMNA (0.83) LMNACYP3A4CYP2D6TSHRRAB9A
Xylazine SCHEMBL22616093 0.90 LMNA (0.81) LMNACYP3A4CYP2D6TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 58450 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260108493-A1 COMPOSITIONS COMPRISING A SEROTONERGIC TRYPTAMINE COMPOUND CAAMTECH, INC. (US) 2026-04-23 US claimed
EP-4727556-A2 SEQUESTRANT COMPOUNDS FOR ALPHA 2 ADRENERGIC AGONISTS Clear Scientific, Inc. (US) 2026-04-22 EP claimed
EP-4724125-A1 APPARATUS, METHODS, AND SYSTEMS FOR ATOMIZED DELIVERY OF A COMPOSITION TO A PATIENT Microneb Tech Holdings, Inc. (US) 2026-04-15 EP claimed
EP-4704826-A1 COMPOSITIONS AND METHODS FOR TREATING POST-TRAUMATIC STRESS DISORDER Yale University (US) 2026-03-11 EP claimed
EP-4704839-A2 IMIDAZOLE CONTAINING COMPOUNDS, DERIVATIVES THEREFORE, AND USES THEREOF ALPHERABIO LLC (US) 2026-03-11 EP claimed
EP-4698287-A1 ANTIMICROBIAL AND DRUG-NEUTRALIZING COMPOSITION SoRite, LLC (US) 2026-02-25 EP claimed
US-20260047623-A1 GLOVE HAVING DRUG-DETECTION COATING SUMMIT GLOVE INC. (US) 2026-02-19 US claimed
WO-2025245294-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USES THEREOF FOR MODULATING WEIGHT GAIN ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245292-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USES THEREOF FOR MODULATING WEIGHT LOSS ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245279-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USE THEREFORE IN TREATMENT OF ADDICTION AND/OR PAIN ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
EP-0220030-B1 ORAL DELIVERY SYSTEM BIOTECHNOLOGY AUSTRALIA PTY. LTD. (AU) 1991-06-19 EP claimed
US-4943428-A 8-HYDROX-2-(DI-N-PROPYLAMINO)TETRALIN WRIGHT STATE UNIVERSITY (US) 1990-07-24 US claimed
US-4921853-A Method for producing analgesia in mammals MICHIGAN STATE UNIVERSITY (US) 1990-05-01 US claimed
CN-86107590-A Oral administration system 1987-05-20 CN claimed
EP-0220030-A2 Oral delivery system BIOTECHNOLOGY AUSTRALIA PTY. LTD. (AU) 1987-04-29 EP claimed
WO-1987002251-A1 ORAL DELIVERY OF BIOLOGICALLY ACTIVE SUBSTANCES BOUND TO VITAMIN B12, OR ANALOGUES THEREOF BIOTECHNOLOGY AUSTRALIA PTY. LTD. (AU) 1987-04-23 WO claimed
US-4614798-A IMPROVED YIELD OF INTERMEDIATE USING TETRAHYDROFURAN OR A MIXTURE OF TOLUENE AND N,N-DIMETHYLACETAMIDE AS SOLVENT VETAMIX (US) 1986-09-30 US claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed
EP-0138358-A1 The preparation and use of 2-[2-(1,4-benzodioxanyl)]-2-imidazoline in therapy Farmos-Yhtyma Oy (FI) 1985-04-24 EP claimed
US-4508715-A DOPAMINE ANTAGONISTS;OVERDOSE TREATMENT UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1985-04-02 US claimed