SCHEMBL15499321

SCHEMBL15499321

COc1ccc(N(c2cccc(OC)c2)c2ccc3c(c2)-c2cc(N(c4ccc(OC)cc4)c4cccc(OC)c4)ccc2-c2ccc(N(c4ccc(OC)cc4)c4cccc(OC)c4)cc2-c2cc(N(c4ccc(OC)cc4)c4cccc(OC)c4)ccc2-3)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 4/20 0.44
HSD17B1 P14061 3/20 0.44
MTNR1A P48039 6/20 0.44
MTNR1B P49286 6/20 0.44
ENPP2 Q13822 1/20 0.43
ALOX15 P16050 1/20 0.41
CYP3A4 P08684 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A1 P04798 1/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP4B1 P13584 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP3A5 P20815 1/20 0.41
CYP2A7 P20853 1/20 0.41
CYP3A7 P24462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8944101 0.91 HSD17B2 (0.50) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL13026514 0.89 CA1 (0.46) ENPP2CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL13385303 0.88 CA4 (0.52) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL12887867 0.88 ABL1 (0.46) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14163837 0.88 ACHE (0.50) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL15497464 0.84 HSD17B2 (0.41) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL8944301 0.84 HSD17B1 (0.51) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL8943967 0.84 HSD17B1 (0.55) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL8820063 0.84 CA4 (0.50) HSD17B2HSD17B1MTNR1AMTNR1BENPP2
SCHEMBL10065629 0.84 CA4 (0.50) HSD17B2HSD17B1MTNR1AMTNR1BENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014037847-A2 NEW SPIRO COMPOUNDS AND THEIR USE IN ORGANIC ELECTRONICS APPLICATIONS AND DEVICES BASF SE (DE) 2014-03-13 WO disclosed
US-20140066656-A1 SPIRO COMPOUNDS AND THEIR USE IN ORGANIC ELECTRONICS APPLICATIONS AND DEVICES BASF SE (DE) 2014-03-06 US disclosed