SCHEMBL15510264

SCHEMBL15510264

CN1CCC(NS(=O)(=O)c2cccc(C3Nc4ccc(OC(=O)O)cc4CC3(C)C)c2)C1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 5/20 0.38
HRH1 P35367 5/20 0.38
NAMPT P43490 1/20 0.37
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
ACHE P22303 4/20 0.34
BCHE P06276 3/20 0.34
HTR1A P08908 5/20 0.34
HTR7 P34969 5/20 0.34
KMT2A Q03164 1/20 0.34
CTSL P07711 1/20 0.34
CTSK P43235 1/20 0.34
DRD2 P14416 1/20 0.34
HTR6 P50406 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2529165 0.89 NAMPT (0.38) HRH2HRH1NAMPTALDH1A1LMNA
SCHEMBL2536830 0.87 HRH2 (0.38) HRH2HRH1NAMPTALDH1A1LMNA
SCHEMBL15510112 0.84 ACHE (0.35) ALDH1A1ACHEBCHE
SCHEMBL15509519 0.81 GFER (0.35) ALDH1A1LMNAACHEBCHE
SCHEMBL15509574 0.81 BRD4 (0.40) ALDH1A1LMNAACHEBCHEKMT2A
SCHEMBL15509834 0.81 GAA (0.42) ALDH1A1LMNAKMT2A
SCHEMBL15509695 0.80 PARP1 (0.38) ACHEBCHEKMT2A
SCHEMBL15509415 0.79 KMT2A (0.36) ALDH1A1LMNAACHEBCHEKMT2A
SCHEMBL15510199 0.78 FAAH (0.41) ACHEBCHE
SCHEMBL15509613 0.77 MCL1 (0.42) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-B1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2014-03-05 EP claimed