SCHEMBL15517474

SCHEMBL15517474

CC(C)(C#C[Si](C)(C)C)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12490127 0.78 ALDH1A1 (0.39) ALDH1A1TSHR
SCHEMBL20158324 0.70 TSHR (0.40) ALDH1A1TSHR
SCHEMBL22532445 0.66
SCHEMBL3956871 0.66
SCHEMBL12372437 0.65 ACLY (0.31) ALDH1A1TSHR
SCHEMBL3533080 0.65 TSHR (0.35) ALDH1A1TSHR
SCHEMBL7064786 0.64
SCHEMBL935231 0.64
SCHEMBL536361 0.61
SCHEMBL1285864 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9790209-B2 Kinase inhibitors RESPIVERT LIMITED (GB) 2017-10-17 US disclosed
US-20160340343-A1 KINASE INHIBITORS OXULAR ACQUISITIONS LIMITED (GB) 2016-11-24 US disclosed
WO-2016109362-A1 CYCLOPROPANECARBOXAMIDE MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR AUSPEX PHARMACEUTICALS, INC. (US) 2016-07-07 WO disclosed
US-20150225373-A1 KINASE INHIBITORS TOPIVERT PHARMA LIMITED (GB) 2015-08-13 US disclosed
EP-2890695-A2 KINASE INHIBITORS Respivert Limited (GB) 2015-07-08 EP disclosed
WO-2014033447-A2 KINASE INHIBITORS RESPIVERT LIMITED (GB) 2014-03-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150225373-A1 KINASE INHIBITORS SYK, SRC, BTK ALDH1A1 2504/4885TSHR 1980/4885
US-20160340343-A1 KINASE INHIBITORS SYK, LYN, BTK ALDH1A1 2404/4885TSHR 2007/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.