SCHEMBL15519637

SCHEMBL15519637

O=C(O)Oc1cccc2[nH]c(-c3ccc(Br)c(F)c3)nc12

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 13/20 0.47
HPSE Q9Y251 1/20 0.45
PARP1 P09874 5/20 0.44
PARP2 Q9UGN5 1/20 0.42
MGAM O43451 1/20 0.41
GAA P10253 1/20 0.41
SI P14410 1/20 0.41
MGAM2 Q2M2H8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15519636 0.82 DHODH (0.70) DHODHPARP1
SCHEMBL15515091 0.79 PARP1 (0.65) DHODHPARP1PARP2
SCHEMBL15520334 0.79 PKN1 (0.63) DHODHPARP1
SCHEMBL6585185 0.76 HPSE (0.44) DHODHHPSEPARP1MGAMGAA
SCHEMBL7861249 0.74 PARP1 (0.53) DHODHHPSEPARP1
SCHEMBL7859132 0.73 PARP1 (0.52) DHODHHPSEPARP1
SCHEMBL7853256 0.73 PARP1 (0.65) DHODHHPSEPARP1
SCHEMBL7860364 0.70 PARP1 (0.69) DHODHPARP1
SCHEMBL7759237 0.70 AURKA (0.54) DHODHHPSEPARP1
SCHEMBL7864193 0.70 PARP1 (0.68) DHODHPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892345-A1 USE OF SUBSTITUTED 2-AMIDOBENZIMIDAZOLES, 2-AMIDOBENZOXAZOLES AND 2-AMIDOBENZOTHIAZOLES OR SALTS THEREOF AS ACTIVE SUBSTANCES AGAINST ABIOTIC PLANT STRESS Bayer CropScience AG (DE) 2015-07-15 EP disclosed
WO-2014037340-A1 USE OF SUBSTITUTED 2-AMIDOBENZIMIDAZOLES, 2-AMIDOBENZOXAZOLES AND 2-AMIDOBENZOTHIAZOLES OR SALTS THEREOF AS ACTIVE SUBSTANCES AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2014-03-13 WO disclosed