SCHEMBL7759237

SCHEMBL7759237

O=C(O)Oc1cccc2[nH]c(-c3ccc(N4CCCC4)nc3)nc12

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.54
AURKB Q96GD4 2/20 0.54
KDR P35968 1/20 0.54
DGAT1 O75907 10/20 0.53
KCNH2 Q12809 8/20 0.53
ADORA2A P29274 7/20 0.53
PARP1 P09874 6/20 0.44
HPSE Q9Y251 1/20 0.42
DHODH Q02127 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
GRIN2B Q13224 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480315 0.99 AURKA (0.53) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL7485013 0.92 AURKA (0.52) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587264 0.91 AURKA (0.55) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587512 0.90 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587278 0.90 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6589042 0.85 AURKA (0.56) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6591285 0.84 AURKA (0.51) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6586056 0.83 AURKA (0.59) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6586837 0.83 AURKA (0.56) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6588365 0.83 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed