SCHEMBL15520366

SCHEMBL15520366

Cn1c(=O)oc2cc(C(C)(c3ccc(-c4ccc(C(=O)O)c(Cl)c4)cc3Cl)C(O)C(F)(F)F)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.44
CMA1 P23946 2/20 0.36
POLB P06746 2/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CTSG P08311 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2C9 P11712 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RORC P51449 1/20 0.33
KMO O15229 1/20 0.33
PDK2 Q15119 1/20 0.33
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
MAPT P10636 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12164118 0.78 CYP11B2 (0.41) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL473809 0.78 CYP11B2 (0.41) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL13183700 0.75 CYP11B2 (0.46) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL12164117 0.72 CYP11B2 (0.39) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL473990 0.72 CYP11B2 (0.39) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL473836 0.72 GPR55 (0.36) CYP11B2POLBKMT2ASMN1; SMN2GPR55
SCHEMBL12164103 0.72 GPR55 (0.36) CYP11B2POLBKMT2ASMN1; SMN2GPR55
SCHEMBL12164182 0.71 CYP11B2 (0.39) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL473871 0.71 CYP11B2 (0.39) CYP11B2CMA1POLBKMT2AALDH1A1
SCHEMBL13183699 0.70 CYP11B2 (0.44) CYP11B2CMA1POLBKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed