SCHEMBL15520801

SCHEMBL15520801

COC(=O)Oc1ccc(-c2ccc(C(C)C(O)(c3ccc4c(c3)N(C)C(=O)CO4)C(F)(F)F)c(Cl)c2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.39
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CTSC P53634 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KMO O15229 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BRD4 O60885 1/20 0.32
USP2 O75604 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
MALT1 Q9UDY8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520373 0.95 GPR55 (0.40) GPR55PDE3BPDE3AMAPTALDH1A1
SCHEMBL15520717 0.94 GPR55 (0.38) GPR55PDE3BPDE3AMAPTALDH1A1
SCHEMBL15520371 0.94 GPR55 (0.37) GPR55PDE3BPDE3AMAPTALDH1A1
SCHEMBL15520843 0.89 GPR55 (0.36) GPR55PDE3BPDE3AMAPTALDH1A1
SCHEMBL15520752 0.89 GPR55 (0.38) GPR55PDE3BPDE3AALDH1A1CTSC
SCHEMBL15520533 0.89 GPR55 (0.38) GPR55PDE3BPDE3AALDH1A1CTSC
SCHEMBL15520803 0.89 GPR55 (0.38) GPR55PDE3BPDE3AALDH1A1CTSC
SCHEMBL12163824 0.89 GPR55 (0.39) GPR55PDE3BPDE3AALDH1A1CTSC
SCHEMBL474432 0.89 GPR55 (0.39) GPR55PDE3BPDE3AALDH1A1CTSC
SCHEMBL15520775 0.88 GPR55 (0.37) GPR55PDE3BPDE3AALDH1A1CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed