SCHEMBL15520775

SCHEMBL15520775

CCOC(=O)Oc1cc(-c2ccc(C(C)C(O)(c3ccc4c(c3)N(C)C(=O)CO4)C(F)(F)F)c(Cl)c2)ccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.37
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BRD4 O60885 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSC P53634 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
KMO O15229 1/20 0.32
SLC5A1 P13866 3/20 0.31
SLC5A2 P31639 3/20 0.31
CUL4A Q13619 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520206 0.91 GPR55 (0.37) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL15520801 0.88 GPR55 (0.39) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL474395 0.88 USP2 (0.37) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL15520717 0.88 GPR55 (0.38) GPR55HTTALDH1A1MEN1KMT2A
SCHEMBL12163847 0.88 USP2 (0.37) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL15520373 0.87 GPR55 (0.40) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL15520371 0.85 GPR55 (0.37) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL15520689 0.85 ALDH1A1 (0.41) USP2HTTL3MBTL1BRD4ALDH1A1
SCHEMBL15520532 0.85 GPR55 (0.38) GPR55USP2HTTL3MBTL1BRD4
SCHEMBL15520843 0.84 GPR55 (0.36) GPR55USP2HTTL3MBTL1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed