SCHEMBL15526231

SCHEMBL15526231

CC(=O)NCCc1cc(Br)ccn1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.50
MTNR1B P49286 6/20 0.50
CYP3A4 P08684 1/20 0.43
PTGFR P43088 1/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
PTGS1 P23219 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
F13A1 P00488 1/20 0.42
ACACB O00763 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15543495 0.84 NPSR1 (0.50) CYP3A4KDM4EALDH1A1MAPTHPGD
SCHEMBL30001281 0.84 NPSR1 (0.50) CYP3A4KDM4EALDH1A1MAPTHPGD
SCHEMBL166146 0.76 ACACB (0.54) MTNR1AMTNR1BKDM4EALDH1A1LMNA
SCHEMBL13605765 0.76 ACACB (0.49) MTNR1AMTNR1BKDM4EALDH1A1LMNA
SCHEMBL48652 0.76 HRH3 (0.61) ALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL12815784 0.75 EGFR (0.46) CYP3A4KDM4EALDH1A1LMNAMAPT
SCHEMBL19783133 0.75 ALDH1A1 (0.41) CYP3A4KDM4EALDH1A1LMNAMAPT
SCHEMBL12815455 0.75 KDM4E (0.41) MTNR1AMTNR1BCYP3A4KDM4EALDH1A1
SCHEMBL1871113 0.75 KDM4E (0.47) CYP3A4KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL19049449 0.74 KDM4E (0.49) MTNR1AMTNR1BCYP3A4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788336-A1 BENZOTHIAZOL- 6 -YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION Gilead Sciences, Inc. (US) 2014-10-15 EP disclosed
WO-2013159064-A1 BENZOTHIAZOL- 6 -YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES, INC. (US) 2013-10-24 WO disclosed