SCHEMBL15526293

SCHEMBL15526293

COC(=O)C(C)(OC(C)(C)C)c1c(C)cc2nc(Br)sc2c1-c1ccc(Cl)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
KDM4E B2RXH2 3/20 0.33
TP53 P04637 2/20 0.33
MDM2 Q00987 2/20 0.33
ALDH1A1 P00352 2/20 0.33
PKM P14618 1/20 0.33
PLA2G2A P14555 1/20 0.33
MAPT P10636 4/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
LCK P06239 1/20 0.32
DHODH Q02127 1/20 0.32
CASP3 P42574 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15526430 0.78 SLC22A12 (0.32) SMN1; SMN2KDM4ENPC1RAB9ADHODH
SCHEMBL15526431 0.78 SLC22A12 (0.32) SMN1; SMN2KDM4ENPC1RAB9ADHODH
SCHEMBL15333587 0.77 CYP3A4 (0.39) SMN1; SMN2L3MBTL1KDM4ETP53MDM2
SCHEMBL15333588 0.77 CYP3A4 (0.39) SMN1; SMN2L3MBTL1KDM4ETP53MDM2
SCHEMBL15331460 0.75 CYP3A4 (0.48) SMN1; SMN2KDM4ENPC1RAB9ASLC22A12
SCHEMBL13735898 0.74 EGFR (0.35) SMN1; SMN2TP53MDM2MAPTNPC1
SCHEMBL19894349 0.74 KMO (0.34) SMN1; SMN2KDM4ENPC1RAB9ASLC22A12
SCHEMBL15331869 0.74 ABL1 (0.39)
SCHEMBL17446789 0.73 CYP3A4 (0.37) L3MBTL1NPC1RAB9ATDP1
SCHEMBL15526296 0.73 CYP3A4 (0.38) SMN1; SMN2L3MBTL1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788336-A1 BENZOTHIAZOL- 6 -YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION Gilead Sciences, Inc. (US) 2014-10-15 EP disclosed
WO-2013159064-A1 BENZOTHIAZOL- 6 -YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES, INC. (US) 2013-10-24 WO disclosed