SCHEMBL15526316

SCHEMBL15526316

CCCCOOC(=O)Cc1c(C)cc2nc(-c3ccc4c(c3)c(-c3cccnc3)nn4C)sc2c1-c1ccc(Cl)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.33
TBXAS1 P24557 1/20 0.33
KDM4E B2RXH2 6/20 0.33
ALDH1A1 P00352 4/20 0.33
HPGD P15428 4/20 0.33
MAPT P10636 4/20 0.33
HSD17B10 Q99714 3/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
TSHR P16473 1/20 0.33
PTGS2 P35354 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
POLB P06746 2/20 0.33
S1PR1 P21453 1/20 0.32
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905916 0.87 KDM4E (0.40) NAMPTTBXAS1KDM4EALDH1A1HPGD
SCHEMBL15526315 0.84 KDM4E (0.34) NAMPTTBXAS1KDM4EALDH1A1HPGD
SCHEMBL15526212 0.83 KDM4E (0.35) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL15526307 0.79 MAPT (0.35) KDM4EALDH1A1HPGDMAPTLMNA
SCHEMBL15342392 0.78 CDC7 (0.35) NAMPTKDM4EALDH1A1HPGDMAPT
SCHEMBL15342020 0.77 CYP3A4 (0.33) NAMPTTBXAS1KDM4EALDH1A1HPGD
SCHEMBL15333463 0.77 CYP3A4 (0.39) NAMPTTBXAS1KDM4EALDH1A1HPGD
SCHEMBL15334233 0.77 CYP3A4 (0.39) NAMPTTBXAS1KDM4EALDH1A1HPGD
SCHEMBL15526288 0.77 KDM4E (0.33) KDM4EALDH1A1HPGDMAPTLMNA
SCHEMBL15526228 0.77 MAPT (0.35) KDM4EALDH1A1HPGDMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788336-A1 BENZOTHIAZOL- 6 -YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION Gilead Sciences, Inc. (US) 2014-10-15 EP disclosed
WO-2013159064-A1 BENZOTHIAZOL- 6 -YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES, INC. (US) 2013-10-24 WO disclosed