SCHEMBL19905916

SCHEMBL19905916

Cc1cc2nc(-c3ccc4c(c3)c(-c3cccnc3)nn4C)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.40
GFER P55789 1/20 0.40
TBXAS1 P24557 1/20 0.39
ALDH1A1 P00352 5/20 0.39
NAMPT P43490 2/20 0.38
MAPT P10636 2/20 0.37
POLB P06746 1/20 0.37
PTGDR2 Q9Y5Y4 4/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
HPGD P15428 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
PTGES2 Q9H7Z7 1/20 0.35
PDE5A O76074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906174 0.89 NAMPT (0.36) KDM4EGFERTBXAS1ALDH1A1NAMPT
SCHEMBL15526316 0.87 NAMPT (0.33) KDM4EGFERTBXAS1ALDH1A1NAMPT
SCHEMBL19906365 0.87 NAMPT (0.38) KDM4EALDH1A1NAMPTPOLBPTGDR2
SCHEMBL19906005 0.86 KDM4E (0.39) KDM4EGFERALDH1A1MAPTPTGDR2
SCHEMBL19905855 0.86 KDM4E (0.39) KDM4EALDH1A1MAPTPOLBPTGDR2
SCHEMBL19905960 0.85 KDM4E (0.42) KDM4EALDH1A1MAPTPOLBPTGDR2
SCHEMBL19906299 0.83 KDM4E (0.44) KDM4EGFERALDH1A1NAMPTMAPT
SCHEMBL15333463 0.83 CYP3A4 (0.39) KDM4EGFERTBXAS1ALDH1A1NAMPT
SCHEMBL15334233 0.83 CYP3A4 (0.39) KDM4EGFERTBXAS1ALDH1A1NAMPT
SCHEMBL19906074 0.83 KDM4E (0.38) KDM4EALDH1A1MAPTPOLBPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed