SCHEMBL15533895

SCHEMBL15533895

COc1ccc(-c2ccnc(Nc3cccc(C(F)(F)F)c3)n2)c(OC)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.58
CDK2 P24941 4/20 0.58
PIK3CG P48736 4/20 0.56
PIK3CA P42336 3/20 0.56
PIK3CB P42338 3/20 0.56
SYK P43405 3/20 0.55
AURKA O14965 3/20 0.55
CDK4 P11802 2/20 0.54
APP P05067 1/20 0.53
ABL1 P00519 2/20 0.53
BCR P11274 1/20 0.53
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
MAPK1 P28482 1/20 0.52
CDK5 Q00535 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
DYRK1B Q9Y463 2/20 0.52
MAP4K4 O95819 1/20 0.52
LCK P06239 1/20 0.52
MET P08581 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15534256 0.85 CCNT1 (0.47) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL15534016 0.81 SYK (0.53) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL15534241 0.81 CLK1 (0.63) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL3247345 0.81 CDK2 (0.56) GSK3BCDK2AURKACDK4ABL1
SCHEMBL27116070 0.79 PIK3CG (0.57) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL12298125 0.79 CSNK2A1 (0.59) GSK3BAPPLMNAMAPTMAPK1
SCHEMBL3257741 0.78 PIK3CG (0.56) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL12274955 0.77 ABL1 (0.56) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL27116137 0.76 GSK3B (0.65) GSK3BCDK2PIK3CGPIK3CAPIK3CB
SCHEMBL25337941 0.76 AURKA (0.62) GSK3BCDK2AURKACDK4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO claimed
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed