SCHEMBL15535452

SCHEMBL15535452

COCCNc1c(C#N)cc(O)c(O)c1C#N.COCCNc1c(C#N)cc(OC)c(OC(=O)OC(C)(C)C)c1C#N

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
DYRK1A Q13627 1/20 0.33
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ENPP1 P22413 1/20 0.31
FGFR4 P22455 3/20 0.31
DNM1 Q05193 1/20 0.31
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
CFTR P13569 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15535829 0.93 ALDH1A1 (0.39) ALDH1A1DYRK1AMEN1KMT2AENPP1
SCHEMBL29391508 0.93 ALDH1A1 (0.39) ALDH1A1DYRK1AMEN1KMT2AENPP1
SCHEMBL29391980 0.88 GAA (0.36) ALDH1A1MEN1KMT2AENPP1KDM4E
SCHEMBL15535973 0.88 GAA (0.36) ALDH1A1MEN1KMT2AENPP1KDM4E
SCHEMBL16969048 0.85 ALDH1A1 (0.43) ALDH1A1DYRK1AMEN1KMT2AENPP1
SCHEMBL15534847 0.81 HTR1A (0.36) ALDH1A1MEN1KMT2AENPP1KDM4E
SCHEMBL29391518 0.81 HTR1A (0.36) ALDH1A1MEN1KMT2AENPP1KDM4E
SCHEMBL15557568 0.80 NSD2 (0.34) ALDH1A1KDM4EGAAHPGD
SCHEMBL16969049 0.80 ALDH1A1 (0.42) ALDH1A1DYRK1AMEN1KMT2AENPP1
SCHEMBL15535447 0.80 ALDH1A1 (0.38) ALDH1A1DYRK1AMEN1KMT2AENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855426-A1 CATECHOL O-METHYLTRANSFERASE ACTIVITY INHIBITING COMPOUNDS Orion Corporation (FI) 2015-04-08 EP disclosed
WO-2013175053-A1 CATECHOL O-METHYLTRANSFERASE ACTIVITY INHIBITING COMPOUNDS ORION CORPORATION (FI) 2013-11-28 WO disclosed