SCHEMBL15535530

SCHEMBL15535530

O=[N+]([O-])c1ccnc(-c2ccc(CCF)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
CES1 P23141 1/20 0.41
KCNH2 Q12809 2/20 0.40
KCNJ1 P48048 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
EIF4A1 P60842 2/20 0.38
NPBWR1 P48145 1/20 0.38
TSHR P16473 1/20 0.38
CYP19A1 P11511 3/20 0.38
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28022013 0.92 FAAH (0.44) FAAHCES1KCNH2KCNJ1CCNC
SCHEMBL545799 0.77 ABL1 (0.53) TSHRCYP19A1CYP11B1CYP11B2LMNA
SCHEMBL826630 0.76 TSHR (0.50) CES1TSHRALDH1A1LMNANPSR1
SCHEMBL1847096 0.74 TSHR (0.64) KCNH2KCNJ1TSHRCYP19A1ALDH1A1
SCHEMBL3133571 0.74 APP (0.51) CDK8TSHRALDH1A1LMNANPC1
SCHEMBL546042 0.71 ABL1 (0.44) FAAHCES1TSHRCYP19A1CYP11B1
SCHEMBL23365096 0.70 NPC1 (0.42) FAAHCES1TSHRALDH1A1LMNA
SCHEMBL546381 0.70 ABL1 (0.59) CYP19A1CYP11B1CYP11B2LMNAMAPT
SCHEMBL29978954 0.70 NPC1 (0.42) FAAHCES1TSHRALDH1A1LMNA
SCHEMBL1816182 0.68 TSHR (0.62) TSHRALDH1A1LMNAMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2852572-A1 CARBOLINE AND CARBAZOLE BASED IMAGING AGENTS FOR DETECTING NEUROLOGICAL DYSFUNCTION Eli Lilly and Company (US) 2015-04-01 EP disclosed
WO-2013176698-A1 CARBOLINE AND CARBAZOLE BASED IMAGING AGENTS FOR DETECTING NEUROLOGICAL DYSFUNCTION ELI LILLY AND COMPANY (US) 2013-11-28 WO disclosed