SCHEMBL15539307

SCHEMBL15539307

COC(=O)c1cccc([N+](=O)[O-])c1NC(C(=O)OC(C)(C)C)c1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
BDKRB1 P46663 1/20 0.36
NPY2R P49146 1/20 0.34
ALDH1A1 P00352 5/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SLC6A3 Q01959 3/20 0.33
SLC6A4 P31645 2/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPK1 P28482 1/20 0.33
F2 P00734 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
BRS3 P32247 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2598198 0.78 BDKRB1 (0.47) BDKRB1ALDH1A1SMN1; SMN2MAPTKDM4E
SCHEMBL31722799 0.78 BDKRB1 (0.47) BDKRB1ALDH1A1SMN1; SMN2MAPTKDM4E
SCHEMBL4939408 0.75 LTB4R2 (0.41) PTPN1GPR119BDKRB1ALDH1A1SMN1; SMN2
SCHEMBL9197575 0.74 L3MBTL1 (0.42) PTPN1BDKRB1ALDH1A1SMN1; SMN2MAPT
SCHEMBL4265981 0.74 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL9192373 0.73 MME (0.38) PTPN1BDKRB1ALDH1A1SMN1; SMN2MAPT
SCHEMBL1421011 0.73 ATR (0.52) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL30063181 0.73 ATR (0.52) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL2598199 0.73 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2SLC6A3SLC6A4MAPT
SCHEMBL3976878 0.72 ALDH1A1 (0.46) BDKRB1ALDH1A1SMN1; SMN2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013186792-A2 PROCESS FOR THE PREPARATION OF (5-METHYL-2-OXO-L,3-DIOXOI-4-VL)METHVL 2- ETHOXV-L-{[2'-(5-OXO-4,5-DIHVDRO-L,2,4-OXADIAZOL-3-VL)BIPHENYI-4-VL]METHYL}- LH-BENZIMIDAZOLE-7-CARBOXYIATE AND ITS SALTS MSN LABORATORIES LIMITED (IN) 2013-12-19 WO disclosed