SCHEMBL15540980

SCHEMBL15540980

CC(C)(C)OC(=O)NC1CC1c1cccc(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.57
MAOB P27338 2/20 0.55
MAOA P21397 1/20 0.51
DPP4 P27487 6/20 0.46
EPHX2 P34913 1/20 0.45
DPP7 Q9UHL4 2/20 0.45
DPP8 Q6V1X1 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TLR2 O60603 1/20 0.43
TLR1 Q15399 1/20 0.43
FAP Q12884 1/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43
SLC9A1 P19634 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15540982 1.00 KDM1A (0.57) KDM1AMAOBMAOADPP4EPHX2
SCHEMBL13272369 0.86 KDM1A (0.58) KDM1AMAOBMAOAEPHX2SMN1; SMN2
SCHEMBL7857682 0.85 KDM1A (0.57) KDM1AMAOBMAOAEPHX2SMN1; SMN2
SCHEMBL21048167 0.85 KDM1A (0.57) KDM1AMAOBMAOAEPHX2SMN1; SMN2
SCHEMBL7904171 0.85 KDM1A (0.57) KDM1AMAOBMAOADPP4DPP8
SCHEMBL15213229 0.84 KDM1A (0.70) KDM1AMAOBMAOADPP4EPHX2
SCHEMBL1570323 0.84 KDM1A (0.70) KDM1AMAOBMAOADPP4EPHX2
SCHEMBL31728997 0.84 KDM1A (0.70) KDM1AMAOBMAOADPP4EPHX2
SCHEMBL4817372 0.84 KDM1A (0.74) KDM1AMAOBMAOAEPHX2SMN1; SMN2
SCHEMBL20724191 0.84 KDM1A (0.74) KDM1AMAOBMAOAEPHX2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2867226-B1 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2018-11-14 EP disclosed
US-9815819-B2 Complement pathway modulators and uses thereof NOVARTIS AG (CH) 2017-11-14 US disclosed
US-9815819-B2 Complement pathway modulators and uses thereof NOVARTIS AG (CH) 2017-11-14 US disclosed
US-20150141455-A1 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2015-05-21 US disclosed
US-20150141455-A1 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2015-05-21 US disclosed
EP-2867226-A2 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF Novartis AG (CH) 2015-05-06 EP disclosed
WO-2014002051-A2 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2014-01-03 WO disclosed
WO-2014002051-A2 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2014-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150141455-A1 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF C5, C3AR1, C9 KDM1A 4705/4885MAOB 265/4885MAOA 412/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.