SCHEMBL15544405

SCHEMBL15544405

O=C1COC2(CCN(Cc3ccc(-c4cccc5ncccc45)cc3F)CC2)CN1C1CC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FASN P49327 6/20 0.49
MLNR O43193 3/20 0.36
ACVR1 Q04771 3/20 0.35
ERN1 O75460 1/20 0.35
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
TYK2 P29597 2/20 0.35
JAK3 P52333 2/20 0.35
OPRM1 P35372 2/20 0.34
OPRK1 P41145 1/20 0.34
CHRM1 P11229 2/20 0.34
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14842076 0.86 FASN (0.65) FASNOPRM1CHRM1SIGMAR1
SCHEMBL15543468 0.86 FASN (0.57) FASNOPRM1CHRM1SIGMAR1
SCHEMBL15544977 0.84 FASN (0.51) FASNACVR1OPRM1CHRM1SIGMAR1
SCHEMBL4542733 0.84 FASN (0.60) FASNACVR1ERN1
SCHEMBL15544087 0.82 FASN (0.48) FASNJAK2TYK2OPRM1OPRK1
SCHEMBL15582390 0.81 FASN (0.60) FASNJAK2OPRM1SIGMAR1
SCHEMBL14720162 0.81 FASN (0.46) FASNACVR1ERN1JAK1JAK3
SCHEMBL15544476 0.81 FASN (0.47) FASNMLNRJAK2JAK1TYK2
SCHEMBL15544497 0.80 FASN (0.42) FASNJAK2TYK2OPRM1OPRK1
SCHEMBL15581938 0.79 FASN (0.49) FASNOPRM1OPRK1CHRM1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO claimed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed