SCHEMBL15544600

SCHEMBL15544600

O=COCc1cc(F)ccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.40
SLC6A4 P31645 5/20 0.40
KCNH2 Q12809 4/20 0.40
SGMS2 Q8NHU3 2/20 0.38
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
SRC P12931 1/20 0.35
HSD11B1 P28845 1/20 0.34
HTR2C P28335 1/20 0.34
IDO1 P14902 2/20 0.34
AGXT P21549 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15544922 0.81 MMP2 (0.42) HTR2ASLC6A4ALDH1A1MEN1POLB
SCHEMBL11308859 0.81 IDO1 (0.40) HTR2ASLC6A4KCNH2SGMS2ALDH1A1
SCHEMBL96253 0.78 IDO1 (0.58) ALDH1A1MEN1POLBHPGDKMT2A
SCHEMBL16545839 0.78 SRC (0.33) HPGDSRC
SCHEMBL16141987 0.76 HTR2A (0.42) HTR2ASLC6A4KCNH2SGMS2HTR2C
SCHEMBL29956098 0.76 HTR2A (0.39) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL9939734 0.76 HTR2A (0.39) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL8184326 0.74 ALDH1A1 (0.48) HTR2ASLC6A4KCNH2ALDH1A1MEN1
SCHEMBL98918 0.73 IDO1 (0.55) HPGDIDO1L3MBTL1
SCHEMBL25292281 0.73 HTR2A (0.38) HTR2ASLC6A4KCNH2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2885307-A1 1-PHENYL-SUBSTITUTED HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS Actelion Pharmaceuticals Ltd. (CH) 2015-06-24 EP disclosed
WO-2014006585-A1 1-PHENYL-SUBSTITUTED HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2014-01-09 WO disclosed