SCHEMBL15548580

SCHEMBL15548580

N#Cc1ccc(O)c(C#N)c1-c1ccccc1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.46
PGR P06401 2/20 0.46
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
ESR2 Q92731 1/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
PIM1 P11309 2/20 0.40
BIRC5 O15392 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
KMT2A Q03164 1/20 0.39
IKBKB O14920 5/20 0.38
HPGD P15428 1/20 0.38
BCL2L1 Q07817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29403248 0.80 ESR2 (0.52) ARPGRMAOAMAOBESR2
SCHEMBL6752587 0.80 ESR2 (0.52) ARPGRMAOAMAOBESR2
SCHEMBL1285853 0.78 ESR2 (0.59) ARPGRMAOAMAOBESR2
SCHEMBL1285672 0.76 ESR2 (0.57) ARPGRMAOAMAOBESR2
SCHEMBL11316898 0.76 ALDH1A1 (0.50) ARPGRMAOAMAOBESR2
SCHEMBL10429209 0.75 ESR2 (0.55) ARPGRMAOAMAOBESR2
SCHEMBL21951910 0.74 PGR (0.43) ARPGRESR2FNTAFNTB
SCHEMBL29692190 0.74 ESR2 (0.46) ARPGRMAOAMAOBESR2
SCHEMBL12679731 0.74 ALDH1A1 (0.46) ARPGRESR2PIM1BIRC5
SCHEMBL30697240 0.74 AR (0.43) ARPGRMAOAMAOBESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855426-A1 CATECHOL O-METHYLTRANSFERASE ACTIVITY INHIBITING COMPOUNDS Orion Corporation (FI) 2015-04-08 EP claimed
WO-2013175053-A1 CATECHOL O-METHYLTRANSFERASE ACTIVITY INHIBITING COMPOUNDS ORION CORPORATION (FI) 2013-11-28 WO claimed