SCHEMBL15548819

SCHEMBL15548819

Cc1nn(C)c(Cl)c1S(=O)(=O)N1CCC(Cc2ccccc2)CC1

nearest known ligand 0.83

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 11/20 0.83
PROKR1 Q8TCW9 11/20 0.83
LMNA P02545 2/20 0.61
TSHR P16473 1/20 0.61
TDP1 Q9NUW8 1/20 0.53
ALDH1A1 P00352 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15549113 0.91 FPR2 (1.00) FPR2PROKR1LMNA
SCHEMBL15548928 0.88 FPR2 (0.79) FPR2PROKR1LMNATSHRALDH1A1
SCHEMBL15549371 0.81 FPR2 (1.00) FPR2PROKR1LMNA
SCHEMBL15549024 0.79 TSHR (0.61) FPR2PROKR1LMNATSHRTDP1
SCHEMBL15549192 0.77 FPR2 (1.00) FPR2PROKR1
SCHEMBL15549025 0.77 TSHR (0.59) FPR2PROKR1LMNATSHRALDH1A1
SCHEMBL31212431 0.75 EBP (0.70) LMNATSHRALDH1A1
SCHEMBL31212435 0.75 EBP (0.70) LMNATSHRALDH1A1
SCHEMBL15548661 0.75 PROKR1 (1.00) FPR2PROKR1
SCHEMBL15536936 0.74 FPR2 (0.58) FPR2PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855449-B1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2018-03-07 EP claimed
EP-2855449-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP claimed
WO-2013179024-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-12-05 WO claimed
EP-2855449-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed
WO-2013179024-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-12-05 WO disclosed