SCHEMBL15549240

SCHEMBL15549240

CC(C)(C)[Si](C)(C)OCC12CC3CC(CC(COc4cc(F)c(C(=O)NS(=O)(=O)N5CCC5)cc4Cl)(C3)C1)C2

nearest known ligand 0.74

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16448665 0.88 SCN9A (0.82) SCN9A
SCHEMBL15535890 0.88 SCN9A (0.84) SCN9A
SCHEMBL15536841 0.86 SCN9A (1.00) SCN9A
SCHEMBL15536840 0.84 SCN9A (0.56) SCN9A
SCHEMBL16389230 0.84 SCN9A (0.96) SCN9A
SCHEMBL16348596 0.80 SCN9A (1.00) SCN9A
SCHEMBL16348628 0.78 SCN9A (1.00) SCN9A
SCHEMBL15536624 0.78 SCN9A (1.00) SCN9A
SCHEMBL15536556 0.78 SCN9A (1.00) SCN9A
SCHEMBL15536324 0.77 SCN9A (1.00) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855428-A1 N-SUBSTITUTED BENZAMIDES AND THEIR USE IN THE TREATMENT OF PAIN Genentech, Inc. (US) 2015-04-08 EP disclosed
WO-2013177224-A1 N-SUBSTITUTED BENZAMIDES AND THEIR USE IN THE TREATMENT OF PAIN GENENTECH, INC. (US) 2013-11-28 WO disclosed