SCHEMBL15550344

SCHEMBL15550344

Cn1cc(-c2cc([N+](=O)[O-])ccc2F)ccc1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
HIF1A Q16665 1/20 0.44
CASP1 P29466 1/20 0.43
CASP3 P42574 1/20 0.43
CASP4 P49662 1/20 0.43
CASP7 P55210 1/20 0.43
CASP9 P55211 1/20 0.43
CASP6 P55212 1/20 0.43
GABRA1 P14867 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
CCKBR P32239 1/20 0.42
GABRA3 P34903 1/20 0.42
OPRK1 P41145 1/20 0.42
MC3R P41968 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
GHSR Q92847 1/20 0.42
PTPRC P08575 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15550056 0.82 HSPB1 (0.56) ALDH1A1GABRA1GABRG2GABRB3GABRA5
SCHEMBL15552702 0.81 HSPB1 (0.55) BRD4
SCHEMBL15551621 0.80 HSPB1 (0.54) ALDH1A1BRD4KMT2AMAPT
SCHEMBL15550839 0.80 BRD4 (0.47) ALDH1A1CASP1CASP3CASP4CASP7
SCHEMBL16791912 0.78 ALDH1A1 (0.42) ALDH1A1HIF1ACASP1CASP3CASP4
SCHEMBL15552065 0.78 BRD4 (0.40) ALDH1A1BRD4CYP3A4TDP1MAPT
SCHEMBL15552160 0.77 BRD4 (0.50) ALDH1A1BRD4KMT2AMAPT
SCHEMBL15551876 0.77 BRD4 (0.50) ALDH1A1BRD4KMT2AMAPTPTGS2
SCHEMBL15551328 0.76 BRD4 (0.46) ALDH1A1HIF1ACASP1CASP3CASP4
SCHEMBL15550329 0.76 BRD4 (0.65) ALDH1A1HIF1AGHSRBRD4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2858990-A1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AbbVie Inc. (US) 2015-04-15 EP disclosed
EP-2858982-A1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AbbVie Inc. (US) 2015-04-15 EP disclosed
WO-2013185284-A1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES ABBOTT LABORATORIES (US) 2013-12-19 WO disclosed
WO-2013188381-A1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES ABBVIE INC. (US) 2013-12-19 WO disclosed