SCHEMBL15564003

SCHEMBL15564003

O=C(O)Cc1ccc(-c2cccc(O)c2)c(F)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.56
AKR1C2 P52895 1/20 0.56
FAAH O00519 1/20 0.52
PTGS2 P35354 1/20 0.52
THRA P10827 1/20 0.47
THRB P10828 1/20 0.47
DGAT1 O75907 1/20 0.46
SOAT1 P35610 1/20 0.46
SELL P14151 2/20 0.46
SELP P16109 2/20 0.46
AKR1B1 P15121 2/20 0.46
LMNA P02545 2/20 0.45
GAA P10253 2/20 0.45
TSHR P16473 2/20 0.45
ABCC4 O15439 1/20 0.45
PTGS1 P23219 1/20 0.45
HTT P42858 1/20 0.45
PLA2G10 O15496 1/20 0.44
PLA2G2A P14555 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Desmethylflurbiprofen SCHEMBL538938 0.86 PTGS1 (0.56) AKR1C3AKR1C2FAAHPTGS2DGAT1
Desmethylflurbiprofen SCHEMBL239447 0.84 PTGS1 (0.55) AKR1C3AKR1C2FAAHPTGS2DGAT1
SCHEMBL15564511 0.83 AKR1C3 (0.51) AKR1C3AKR1C2FAAHPTGS2LMNA
SCHEMBL4943055 0.83 CA2 (0.56) FAAHPTGS2THRATHRBDGAT1
Methane SCHEMBL11691361 0.82 CA2 (0.55) FAAHPTGS2THRATHRBDGAT1
SCHEMBL4945342 0.80 CA2 (0.56) DGAT1SOAT1AKR1B1LMNAGAA
SCHEMBL3914326 0.79 GRIA2 (0.59) PTGS2THRATHRBAKR1B1LMNA
SCHEMBL31225628 0.79 GRIA2 (0.59) PTGS2THRATHRBAKR1B1LMNA
SCHEMBL6564239 0.78 ABCC4 (0.69) AKR1B1LMNAGAATSHRABCC4
SCHEMBL3642916 0.77 AKR1C3 (0.59) AKR1C3AKR1C2LMNAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2880015-B1 MULTITARGET FAAH AND COX INHIBITORS AND THERAPEUTICAL USES THEREOF FOND ST ITALIANO TECNOLOGIA (IT) 2017-09-27 EP disclosed
EP-2880015-A1 MULTITARGET FAAH AND COX INHIBITORS AND THERAPEUTICAL USES THEREOF Fondazione Istituto Italiano Di Tecnologia (IT) 2015-06-10 EP disclosed
WO-2014023643-A1 MULTITARGET FAAH AND COX INHIBITORS AND THERAPEUTICAL USES THEREOF FONDAZIONE ISTITUTO ITALIANO DI TECNOLOGIA (IT) 2014-02-13 WO disclosed
WO-2014023325-A1 MULTITARGET FAAH AND COX INHIBITORS AND THERAPEUTICAL USES THEREOF FONDAZIONE ISTITUTO ITALIANO DI TECNOLOGIA (IT) 2014-02-13 WO disclosed