SCHEMBL4945342

SCHEMBL4945342

O=C(O)Cc1ccc(-c2ccc(O)cc2F)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.56
CAMK2A Q9UQM7 1/20 0.56
HCAR2 Q8TDS4 2/20 0.52
DGAT1 O75907 2/20 0.52
SOAT1 P35610 2/20 0.52
ESR1 P03372 1/20 0.51
ESR2 Q92731 1/20 0.51
PSEN1 P49768 1/20 0.50
PSEN2 P49810 1/20 0.50
APH1B Q8WW43 1/20 0.50
NCSTN Q92542 1/20 0.50
APH1A Q96BI3 1/20 0.50
PSENEN Q9NZ42 1/20 0.50
AKR1B1 P15121 2/20 0.49
ABCC4 O15439 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
TSHR P16473 1/20 0.49
PTGS1 P23219 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4943055 0.90 CA2 (0.56) CA2CAMK2AHCAR2DGAT1SOAT1
Methane SCHEMBL11691361 0.89 CA2 (0.55) CA2CAMK2AHCAR2DGAT1SOAT1
SCHEMBL11466357 0.85 PPARG (0.56) CA2DGAT1SOAT1PSEN1PSEN2
SCHEMBL5537352 0.82 CYP4F2 (0.50) HCAR2ESR1ESR2GAAAPP
SCHEMBL4943262 0.81 HSD17B1 (0.59) CA2CAMK2AHCAR2DGAT1SOAT1
SCHEMBL1678991 0.81 CA2 (0.56) CA2CAMK2AHCAR2DGAT1SOAT1
SCHEMBL15564003 0.80 AKR1C3 (0.56) CA2CAMK2ADGAT1SOAT1PSEN1
Desmethylflurbiprofen SCHEMBL538938 0.80 PTGS1 (0.56) DGAT1SOAT1PSEN1PSEN2APH1B
Desmethylflurbiprofen SCHEMBL239447 0.79 PTGS1 (0.55) DGAT1SOAT1PSEN1PSEN2APH1B
SCHEMBL38659424 0.78 ESR1 (0.70) ESR1ESR2APPCYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080004301-A1 Benzene Compound Having 2 or More Substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-01-03 US disclosed
EP-1806332-A1 BENZENE COMPOUND HAVING 2 OR MORE SUBSTITUENTS Daiichi Sankyo Company, Limited (JP) 2007-07-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004301-A1 Benzene Compound Having 2 or More Substituents NR1H2, NR1H3, NCOR2 CA2 4239/4885CAMK2A 2270/4885HCAR2 437/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.