SCHEMBL15565149

SCHEMBL15565149

O=c1[nH]c(=O)n(CCc2ccccc2O)nc1O

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DAO P14920 8/20 0.58
HRH3 Q9Y5N1 3/20 0.42
CYP1A2 P05177 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
CYP2C19 P33261 1/20 0.35
HSPA5 P11021 1/20 0.34
AKR1B1 P15121 1/20 0.34
MPO P05164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15565182 1.00 DAO (0.58) DAOHRH3CYP1A2TAAR1CYP2C19
SCHEMBL15564051 0.87 DAO (0.57) DAOTAAR1
SCHEMBL15563911 0.86 DAO (0.56) DAOCYP1A2TAAR1CYP2C19
SCHEMBL15564169 0.84 DAO (0.57) DAO
SCHEMBL15563710 0.83 DAO (0.58) DAOHRH3CYP1A2TAAR1CYP2C19
SCHEMBL15564271 0.82 DAO (0.55) DAO
SCHEMBL15565204 0.81 DAO (0.50) DAO
SCHEMBL15564747 0.80 DAO (0.49) DAOCYP1A2CYP2C19
SCHEMBL15565177 0.80 DAO (0.49) DAO
SCHEMBL15564237 0.78 DAO (0.58) DAOCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9505753-B2 Inhibitors of D-amino acid oxidase THE JOHNS HOPKINS UNIVERSITY (US) 2016-11-29 US claimed
US-20150218156-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2015-08-06 US claimed
WO-2014025993-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2014-02-13 WO claimed
US-9505753-B2 Inhibitors of D-amino acid oxidase THE JOHNS HOPKINS UNIVERSITY (US) 2016-11-29 US disclosed
US-20150218156-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2015-08-06 US disclosed
WO-2014025993-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2014-02-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150218156-A1 INHIBITORS OF D-AMINO ACID OXIDASE DDO, DAO, GRIN2A DAO 2/4885HRH3 1538/4885CYP1A2 2331/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.