SCHEMBL15567959

SCHEMBL15567959

CC(=O)N1CCN(CCCc2nc3ccccc3n2Cc2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 4/20 0.56
AGTR2 P50052 4/20 0.56
POLB P06746 2/20 0.53
ALDH1A1 P00352 6/20 0.53
MEN1 O00255 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
DRD2 P14416 1/20 0.52
DRD4 P21917 1/20 0.52
DRD3 P35462 1/20 0.52
ALDH1A2 O94788 4/20 0.52
ALDH2 P05091 4/20 0.52
ALDH3A1 P30838 4/20 0.52
ALDH1A3 P47895 4/20 0.52
PPARG P37231 3/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15568517 0.88 ALDH1A1 (0.69) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL15568680 0.87 MEN1 (0.60) AGTR1AGTR2ALDH1A1MEN1CYP1A2
SCHEMBL15568703 0.83 MEN1 (0.72) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL16556627 0.78 MEN1 (0.60) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL13187162 0.77 HIF1A (0.76) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL15568343 0.76 ALDH1A1 (0.67) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL9740603 0.75 ALDH1A1 (0.66) AGTR1AGTR2POLBALDH1A1MEN1
SCHEMBL6213576 0.75 PDE4A (0.69) POLBALDH1A1MEN1KMT2A
SCHEMBL16556624 0.75 MEN1 (0.59) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL229324 0.74 MEN1 (0.78) AGTR1AGTR2POLBALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed