SCHEMBL15568517

SCHEMBL15568517

CC(=O)N1CCN(Cc2nc3ccccc3n2Cc2ccccc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.69
CYP1A2 P05177 2/20 0.69
CYP2D6 P10635 2/20 0.69
CYP2C9 P11712 2/20 0.69
CYP2C19 P33261 2/20 0.69
MEN1 O00255 2/20 0.69
KMT2A Q03164 2/20 0.69
ALDH1A2 O94788 7/20 0.64
ALDH2 P05091 7/20 0.64
ALDH3A1 P30838 7/20 0.64
ALDH1A3 P47895 7/20 0.64
GRM2 Q14416 1/20 0.59
HIF1A Q16665 2/20 0.58
TDP1 Q9NUW8 2/20 0.58
NR1I2 O75469 1/20 0.58
ABCB11 O95342 1/20 0.58
LMNA P02545 1/20 0.58
ESR1 P03372 1/20 0.58
PGR P06401 1/20 0.58
CYP3A4 P08684 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15567959 0.88 AGTR1 (0.56) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15568343 0.87 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15569151 0.84 FAAH (0.66) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15567214 0.84 ALDH1A1 (0.63) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15568741 0.84 ALDH1A1 (0.63) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15568555 0.84 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15569377 0.82 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15568468 0.81 MEN1 (0.74) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
Clemizole SCHEMBL19976081 0.81 HIF1A (0.84) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL28991317 0.81 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed