SCHEMBL15569007

SCHEMBL15569007

CC(C)(C(=O)O)c1ccc(CCN2CCC(c3nc4ccccc4n3C3CO3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 10/20 0.55
OPRL1 P41146 4/20 0.45
OGFRL1 Q5TC84 4/20 0.45
HRH3 Q9Y5N1 1/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
KCNH2 Q12809 2/20 0.42
TACR2 P21452 1/20 0.42
TACR1 P25103 1/20 0.42
LMNA P02545 1/20 0.42
CNR1 P21554 1/20 0.42
APEX1 P27695 1/20 0.42
PDE4A P27815 1/20 0.42
HTR2A P28223 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2B P41595 1/20 0.42
BLM P54132 1/20 0.42
PDE3A Q14432 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13624817 0.89 HRH1 (0.58) HRH1HRH3USP2POLBKCNH2
SCHEMBL4653613 0.86 HRH1 (0.63) HRH1HRH3USP2POLBKCNH2
SCHEMBL18884525 0.84 HRH1 (0.68) HRH1USP2POLBKCNH2TACR2
Bilastine SCHEMBL29402994 0.82 HRH1 (0.82) HRH1USP2POLBKCNH2
Bilastine SCHEMBL991810 0.82 HRH1 (0.82) HRH1USP2POLBKCNH2
Bilastine SCHEMBL21815518 0.80 HRH1 (0.77) HRH1KCNH2LMNA
SCHEMBL993093 0.77 HTR2B (0.55) HRH1POLBKCNH2TACR2HTR2B
SCHEMBL11977258 0.75 HRH1 (0.72) HRH1KCNH2LMNACNR1APEX1
SCHEMBL991771 0.74 HRH1 (0.79) HRH1KCNH2
SCHEMBL3793927 0.74 HRH1 (0.79) HRH1KCNH2TACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014026657-A2 A PROCESS FOR THE PREPARATION OF A DERIVATIVE OF 2-METHYL-2'-PHENYLPROPIONIC ACID USING NEW INTERMEDIATES ZENTIVA, K.S (CZ) 2014-02-20 WO claimed