SCHEMBL15569064

SCHEMBL15569064

O=C(N(CCc1ccccc1)c1ccc(-c2nc3ccccc3n2Cc2ccccc2)cc1)C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
PDE6D O43924 4/20 0.56
ALDH2 P05091 1/20 0.56
ALDH3A1 P30838 1/20 0.56
TP53 P04637 4/20 0.51
HTT P42858 3/20 0.51
MAPT P10636 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HPGD P15428 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
BRD4 O60885 3/20 0.48
DRD2 P14416 1/20 0.47
TBXA2R P21731 1/20 0.47
KDM4E B2RXH2 3/20 0.47
LMNA P02545 2/20 0.47
CNR2 P34972 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HSD17B10 Q99714 1/20 0.46
CFTR P13569 1/20 0.45
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15567143 0.95 ALDH1A1 (0.58) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15568525 0.90 ALDH1A1 (0.55) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15568648 0.90 ALDH1A1 (0.61) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15569562 0.87 ALDH1A1 (0.52) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15568320 0.84 ALDH1A1 (0.70) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15568269 0.84 ALDH1A1 (0.57) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15567956 0.83 ALDH1A1 (0.52) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15567574 0.82 DRD2 (0.51) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15568475 0.81 ALDH1A1 (0.53) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15569279 0.80 ALDH1A1 (0.57) ALDH1A1PDE6DALDH2ALDH3A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed